Thiethylperazine
Thiethylperazine (Torecan) is an antiemetic of the phenothiazine class. Though it was never licensed or used as an antipsychotic, it may have such effects.
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| AHFS/Drugs.com | Micromedex Detailed Consumer Information |
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| Protein binding | 60% |
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| ECHA InfoCard | 100.014.381  |
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| Formula | C22H29N3S2 |
| Molar mass | 399.62 g·mol−1 |
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Thiethylperazine activates the transport protein ABCC1 that clears beta-amyloid from brains of mice.[1]
References
- Krohn M, Lange C, Hofrichter J, Scheffler K, Stenzel J, Steffen J, et al. (October 2011). "Cerebral amyloid-β proteostasis is regulated by the membrane transport protein ABCC1 in mice". The Journal of Clinical Investigation. 121 (10): 3924–31. doi:10.1172/JCI57867. PMC 3195473. PMID 21881209. Lay summary – Science Daily.
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